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 Benzene ring
 Heterocycles
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Products
 5-Hydroxyisoquinoline
 2-pyridylacetone
 4-Pyrimidinecarboxylic acid, 1,6-dihydro-2-methyl-6-oxo-
 3-FLUORO-2-NITROBENZOIC ACID
 2-Pyridinemethanol, 4-amino-
 2-(HYDROXYMETHYL)ACRYLICACIDETHYLESTER
 3-AMINO-4-BROMOPHENOL
 2-(2,4-Dichlorophenoxy)acetamidine hydrochloride
 1-Methyl-3-(trifluoromethyl)-1H-pyrazol-4-amine
 methyl 4-(1-aminocyclopropyl)benzoate hydrochloride
 4-Fluoro-3-[(trifluoromethyl)sulfonyl]benzenesulfonamide
 6-Quinolinecarboxylic Acid
 5-fluoro-2-methoxypyrine-4-boronic acid
 3,6-Dihydro-2H-pyran-4-carbonitrile
 1-Methyl-1H-indazol-3-carbonyl chloride
 2-fluoro-N-methyl Benzeneethanamine HCL
 Methyl 4-Benzyl-5-oxomorpholine-3-carboxylate
 EthylMorpholine-2-carboxylate
 2,2-dimethyl-N-(2-oxo-3-piperidinyl)Propanamide
 N-(2-amino-4-methylpentyl)Carbamic acid 1,1-dimethylethyl ester
 4-CHLORO-5-FLUORO-2-PYRIDINEMETHANOL
 3-Fluorodibenz[b,e]oxepin-11(6H)-one
 5-Bromo-2,3-dihydro-7-azaindole
 5-ACETYL-2-AMINO-4-HYDROXYBENZOIC ACID
 ETHYL 4-(TRIFLUOROMETHYL)-2-METHYLTHIAZOLE-5-CARBOXYLATE
 tert-butyl 6-oxo-2,7-diazaspiro[4.4]nonane-2-carboxylate
 Imidazo[1,5-a]pyridine-1-carboxylic acid, ethyl ester
 3-Chloro-6-chloromethylpyridazine
 2-Methyl-3-phenoxybenzaldehyde
 2-(5-Aminopyridin-2-yl)-2-methylpropanenitrile
 (R)-1-Benzyl-3-dimethylaminopyrrolidine Dihydrochloride
 EthylImidazo[1,2-a]pyridine-3-carboxylate
 6-bromo-3-iodo-Imidazo[1,2-a]pyrazine
 4-(Bromomethyl)tetrahydropyran
 4-Chloro-6,7-dihydro-5H-cyclopenta[b]pyridin-7-ol
 6-Ethyl-3-pyridinamine
 tert-Butyl 2-methylhydrazinecarboxylate
 METHYLOCTAHYDROPYRROLO[3,4-B]PYRROLE
 6-Benzyl-1H-octahydropyrrolo[3,4-b]pyridine
 2-Chloro-1-methylimidazole-5-boronicAcid Pinacol Ester
 1-BENZYL-OCTAHYDRO-PYRROLO[3,4-B]PYRROLE
 (R)-(+)-3-(Dimethylamino)pyrrolidine
 5-Hydroxy-2-methylindole
 4,6-dichloro-5-nitropyrimidin-2-amine
 4-Nitropyridine-2-carboxylic Acid
 (3aR,6aR)-1-Methyl-hexahydropyrrolo[3,4-b]pyrrole
 2,4-DICHLORO-5-IODOPYRIMIDINE
 1H-Pyrrolo[2,3-b]pyridine-2-carboxylicAcid
 (R)-2-(3-Fluorophenyl)pyrrolidine L-Tartrate
 (R)-7-methyl-1,4-oxazepane hydrochloride
Lead optimization

Our Chemistry Department has extensive expertise and successful track records in early stage drug discovery including hit identification, hit to lead optimization and lead selection, as well as optimization, for the discovery of small-molecule drugs.

Teams utilize both combinatorial and traditional approaches to optimize lead compounds for structure-activity relationships studies by leveraging our vast medicinal chemistry knowledge. Further, our teams can design and synthesize advanced leads to optimize potency, selectivity and specificity, and deliverability to provide your candidate.


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